本书介绍了目前全球正在临床研究中的小分子抗癌新药，它们中的一些将会在今后20年内逐步成为人类战胜癌症的新武器。本书从一个侧面反映出人类目前抗癌新药研发的总体水平和现状。本书以药物名称为序，并包含了下列条目：药物名称、中文参考译名、其他名、研究开发机构、化学结构、当前临床研究进展、药物简介、类似活性化合物及参考文献等。此外，本书还在相关条目下，通俗易懂地介绍了当今国际小分子抗癌药物研究领域中的各种新成果、新理论、新技术和新的发展趋势。本书共包含了小分子抗癌候选药物384个，类似结构的活性化合物4000多个。
本书适合于药学专业和有机化学专业、生物制药专业的教学、科研、管理和情报人员，癌症相关的基础与临床研究人员，从事客户委托药物研发业务的科研人员阅读。
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目录
- 2DG
A-007
Abiraterone acetate
ABT-518
ABT-751
ABT-869
ABT-888
Acadesine
Acetylcysteine
AEE788
AEZS-108
AEZS-112
Afimoxifene
Alanosine
ANA773
Apaziquone
Aplidine
ALS-357
Alvespimycin
Alvocidib
Amifostine
Amonafide dihydrochloride
Amonafide maleate
Amrubicin
Anamorelin hydrochloride
Annamycin
ANX-510
AP5346
AP24534
APO866
Aroplatin
ARQ 197
ARRY-334543
ARRY-142886
Arzoxifene
AT-101
AT7519
Atamestane
Atiprimod
ATN-161
ATN-224
Atrasentan
AVE 8062
AVN-944
Axitinib
AZD0503
AZD1152
AZD 2281
AZD 5896
Banoxantrone
Batabulin sodium
Becatecarin
Belinostat
Bendamustine
Beraprost
Berubicin
BIBW 2992
Bleomycin
BMS-275183
BMS-599626
BN 2629
BN 83495
Bosutinib
Brivanib alaninate
Brostallicin
BSI-201
BZL101
Calcitriol
Canertinib
Canfosfamide
Carbendazim
Carfilzomib
Carmustine
Casopitant mesylate
CBP 501
CC-8490
CDB-4124
Cediranib
Celecoxib
Cemadotin
CEP-7055
Cevipabulin fumarate
CF 101
CGC-11047
CHIR-258
CHIR-265
Chlorpromazine and pentamidine
Cilengitide
Clodronic acid
CNF-2024
Combretastatin A-4 phosphate
CP-547632
CP-724714
CP-868596
CRA-024781
CS-7017
CT-2106
Darinaparsin
Deforolimus
Degarelix
Demethylpenclomedine
Denibulin
Diethylnorspermine
Dexmethylphenidate hydrochloride
DHA-paclitaxel
Diflomotecan
Dimesna
DJ-927
DMXAA
Docosahexaenoic acid
Doxorubicin
Doxorubicin inhaled
Doxorubicin liposomal
Dutasteride
E 7080
E 7820
E 7974
EC 0225
EC17
EC20
EC145
Edatrexate
Edotecarin
Edotreotide
Efaproxiral
Elacridar
Elagolix
Elinafide
Elsamitrucin
Elesclomol
Eltrombopag
Eniluracil
ENMD-1198
Enzastaurin
EPC 2407
Epothilone D
Eribulin mesylate
ES-285
Etalocib
Ethonafide
Ethynylcytidine
Exatecan
Exherin
Ezatiostat hydrochloride
Fentanyl
Fentanyl inhalation
Fentanyl intranasal
Fentanyl transmucosal
Fludarabine
Forodesine
Gallium maltolate
Gefitinib
Gimatecan
Glufosfamide
Glutamine
Goserelin
Gossypol
GPX-100
GPX-150
Hexyl 5-aminolevulinate
Histamine
HKI-272
HMN-176
HMN-214
Omacetaxine mepesuccinate
IDM-2101
Imexon
Imidazoacridone
INCB 7839
Indibulin
Indisulam
INNO-206
INNO-305
INNO-406
INO-1001
INSM-18
Iobenguane
Irofulven
Isatoribine
Ispinesib
Ixabepilone
JNK 401
Kahalalide F
Karenitecin
Ketamine
KOS-1584
KOS-1584
KRX-0402
KRX-0601
L-377202
Lanreotide
Laromustine
Larotaxel
Lasofoxifene
LE-SN38
Lestaurtinib
Levoleucovorin
Lomeguatrib
Lonafarnib
LR-103
Lucanthone
LY-573636
M 40403
MB 07133
MDAM
Incyclinide
2-methoxyestradiol
MGCD-0103
MGCD265
Midostaurin
Mifamurtide
Mifepristone
Milataxel
Miltefosine
MIP-1104
MK-0457
MK-0731
MK-0752
MKC-1
MLN2238
MLN8054
MLN8237
Morphine intranasal
Morphine intranasal（RylomineTM）
Motexafin gadolinium
MP-470
MPC-2130
MPC-6827
NAC
NBI 42902
Nilotinib
NM-3
Nolatrexed
Noscapine
NOV-002
NPI 2358
Obatoclax
Octreotide（Atrigel®）
Octreotide（Sandostatin®）
Oleandrin
ON 01910
Ortataxel
OSI-906
OSI 930
Oxycodone and naltrexone
Ozarelix
P2045
Paclitaxel（LEP-ETU）
Paclitaxel（OncoGel）
Paclitaxel（AI 850）
Paclitaxel poliglumex
Paclitaxel（Tocosol）
Palifosfamide
Palonosetron
Pamidronic acid
Patupilone
PCK 3145
PCI-24781
PCI-27483
PCI-32765
Phenoxodiol
Pralatrexate
Pelitinib
Pelitrexol
PEP-005
Perifosine
PHY 906
Picoplatin
Pipendoxifene
Pixantrone
Plerixafor
Plevitrexed
Plitidepsin
PM00104
PM02734
Pomalidomide
PPI 2458
PX-12
PX-478
PX-866
Pyroxamide
Quarfloxin
Quinagolide
R547
R1645
R1668
RC-3095
Relacatib
Retaspimycin
RH1
Romidepsin
Ropidoxuridine
Roquinimex
Rosabulin
RP101
RTA 402
Rubitecan
S-1
Salinosporamide A
Sapacitabine
Satraplatin
SB-743921
Seliciclib
Semapimod
Seocalcitol
Silibinin
Simotaxel
SN-2310
SNS-032
SNS-314
SNS-595
Sodium phenylbutyrate
Sodium stibogluconate
SPI-1620
Squalamine lactate
SR 31747
STA-9090
Sodium thiosulfat
SU14813
TAC-101
Talabostat
Talampanel
Talaporfin sodium
Taltobulin
Talotrexin Ammonium
Tamibarotene
Tandutinib
Tanespimycin
Tarenflurbil
Tariquidar
TAS-102
TAS-108
Tasidotin hydrochloride
Tegafur and uracil
Temsirolimus
Terameprocol
Tesmilifene
Tetrandrine
Thymalfasin
Thymectacin
Tipifarnib
Tirapazamine
Telatinib
TL-310
TPI 287
Trabectedin
Tretazicar
Tretinoin
Triapine
Triciribine
Trilostane
Troxacitabine
TSU-68
TXD-258
UCN-01
Ukrain
Uracil
Uridine triacetate
Vandetanib
Vatalanib succinate
Verteporfin
Vincristine sulfate
Vincristine tartrate
Vinflunine
VX944
WF10
WX-671
WX-UK1
Xaliproden
XL019
XL147
XL184
XL228
XL281
XL581
XL647
XL765
XL820
XL844
XL880
YM155
ZD4054
ZK-epothilone
Zosuquidar trihydrochloride
附录1 抗癌新药化学结构索引
附录2 抗癌新药按作用机制分类索引
附录3 抗癌新药按研发厂商名索引
附录4 活性化合物按取代基索引
附录5 活性化合物按母体化学结构索引
附录6 新技术、新理论和研究专题索引
附录7 中文总索引
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